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Acanthaceae: a family of medicinal plants

Classification

Kingdom  Plantae – Plants
Subkingdom  Tracheobionta – Vascular plants
Superdivision  Spermatophyta – Seed plants
Division  Magnoliophyta – Flowering plants
Class  Magnoliopsida – Dicotyledons
Subclass  Asteridae
Order  Scrophulariales

Family  Acanthaceae – Acanthus family

Introduction

This family is a main group of flowering plants also termed as Angiosperms containing more than 2500 species classified into more than 200 genera. Most of them are shrubs, tropical herbs or twining vines.  Plants belonged to Acathaceae are mainly located in Brazil, Africa, Central America, Malaysia and  Indonesia. These plants are found in open forests, dense forests, wet fields, valleys, marine areas, mangrove forests, scrublands and sea coast area. In short they are found in every place.  
Acanthaceae has few worldwide features present in its species. Majority of them have simply arranged in opposite pairs of leaves, with crystals of calcium carbonate in protuberances or streaks in the vegetative parts. They have bisexual flowers with bilaterally symmetry and mostly enclosed by large and colored leaflike bracts.  Petals and sepals are four or five in number which are frequently fused into tubular structures. Acanthaceae usually have two or four stamens, extending outside the flower mouth frequently with one- three sterile stamens or staminodes. The pistil is superior means they are positioned above the attachment point of the other flower parts and commonly contains two fused ovule-bearing segments enclosing two chambers.  Each of these contains two-much ovules in the form of two rows along the central axis of the ovary. 


Importance:

The major economic importance of the family is horticultural. Species of Acanthus, Odontonema Nees, Aphelandra R. Brown, Crossandra Salisbury, Thunbergia,  Barleria , Eranthemum, Pachystachys Nees,  Justicia, Ruellia, Sanchezia Ruiz & Pavon, Fittonia, and various other genera are extensively cultivated as ornamentals. Many species are cultivated in and Pakistan. These include: Barleria lupulina Lindley, Aphelandra squarrosa Nees, Sanchezia parvibracteata Sprague & Hutchinson, Eranthemum pulchellum Andrews, Fittonia albivenis (Veitch) Brummitt, Thunbergia erecta (Bentham) T. Anderson,  Justicia betonica Linnaeus, J. brandegeeana Wasshausen & L. B. Smith, J. carnea Lindley, Pachystachys lutea Nees, Ruellia elegans Poiret, Crossandra infundibuliformis (Linnaeus) Nees,  R. simplex C. Wright,  and T. laurifolia Lindley.


Ethnomedicinal Uses:

Plants belong to Acanthaceae are also medicinal important. For example Blepharis maderaspatensis leaves are mixed with onion bulb to form a paste and it is externally applied to wounds and cuts. Leaves of Justicia tranquebariensis are used for poisonous bites and Hygrophila auriculata leaves for cough relieve. Leaves of Asystasia schimperi, Dyschoriste thumbergiiflora, Dyschoriste radicans, Lepidagathis scariosa, Acanthus eminens, Thunbergia alata are used to make an infusion to cure cough, eye infections,  skin disease, anti-diarrhea,  wounds, edema,  backache and pneumonia. Ash of leaves of Justicia  betonica,  Acanthus pubescens and Justicia  flava is used for dry cough, ulcer, anti-diarrhea and flu. Leaves of Justicia adhatoda are used for chest disease, rheumatism, fever, asthma, pneumonia, tuberculosis, diuretic, antispasmodic, antiseptic, expectorant, and to reduce swelling. Blepharis maderaspatensis,  Andrographis  paniculata, Elytraria acualis are used externally for wounds, internally for diabetes and externally for hip pain respectively.


Pharmacological Activities:

Plants of Acanthaceae family have showed significant antibacterial activity against Escherichia coli, Staphylococcus aereus, Bacillus subtilis, Pseudomonas aeruginosa, Proteus vulgaris and Klebsiella pneumoniae. Among many tested plant against bacterial strains, chloroform crude extract of Andrographis paniculata showed remarkable antibacterial activity comparable to many antibiotics. Hypoestes Serpens, Andrographis paniculata, Rhinacanthus nasutus are antiviral plants agaisnt a wide range of fungal species.
Other pharmacological activities which belong to Acanthaceae are cytotoxicity, antioxidant, anti inflammatory, antipyretic activity, hepatoprotective activity, insecticidal activity, immunomodulatory activity and antiplatelet aggregation activity.


Phytochemistry:

Phytochemical reports on family Acanthaceae are glycosides, benzonoids, flavonoids, phenolic compounds, triterpenoids,  naphthoquinone.

Glycosides:
  • (2R)-2-O-β-D-gluco-pyranosyl-2H-1,4- benzoxazin-3(4H)-one,
  • (2R)-2-O-β-D-glucopyranosyl-4- hydroxy-2H-1,4-benzoxazin-3(4H)–one,
  • (2R)-2-O-β- D-glucopyranosyl-7-hydroxy-2H-1,4-benzoxazin-3(4H)-one,
  • 7- chloro-(2R)-2-O-β-D-glucopyranosyl-2H-1,4-benzoxazin-3(4H)-one,
  • (2R)-2-O-β-D-glucopyranosyl-5-hydroxy-2H-1,4- benzoxazin-3(4H)-one,
  • benzyl β-D-glucopyranoside,
  • apigenin 7-O-β-D-glucopyranoside,
  • apigenin 7-O-neohesperidoside,
  • apigenin 7-O-β-Dglucopyranosy (1→ 6) -β-D-glucopyranoside,
  • Olean-12-ene-1β,3β,11α,28-tetraol-28-O-β-D-glucopyranosyl-(1→2) -β-D-glucopyranoside,
  • olean-12-ene-1β,3β,11α,28-tetraol-28- O-β-D-glucopyranosyl-(1→2)-β-D-glucopyranosyl-(1→2)-β-D-gluco pyranoside,
  • 11α-methoxy-olean-12-ene-1β,3β,28-triol-28-O-β- D-glucopyranosyl-(1→2)-β-D-glucopyranoside,
  • 11α- methoxy-olean-12-ene-1β, 3β, 28-triol 28-O-β-Dglucopyranosyl- 1→2)-β-D-glucopyranosyl-(1→2)-β-D-glucopyranoside,
  • Salidroside, ajugol, desrhamnosylacteoside, poliumoside, acteoside, verbascoside, decaffeoylverbascoside, isoverbascoside, leucosceptoside A, ebracteatoside B, angeloside and Luteolin7-O-β-D-glucopyranoside


Naphthoquinone
Following Naphthoquinones are present in acanthaceae: Rhinacanthin A, rhinacanthin B, rhinacanthin C, rhinacanthin D, rhinacanthin G, rhinacanthin H, rhinacanthin I, rhinacanthin J, rhinacanthin K, rhinacanthin L, rhinacanthin M, rhinacanthin N, rhinacanthin O, rhinacanthin P and rhinacanthin Q. While Rhinacanthins showed remarkable cytotoxic, antiviral and antiplatelet aggregation activity.

Flavonoids
3-epi-ursolic acid, verbascoside, andrographolide, sitosterol, 7-O-methyldihydrowogonin, dihydroskullcapflavone I, 5-hydroxy-7,8,2’,5’-tetramethoxy-flavone, skullcapflavone12’- methylether, chlorogenic acid, 7-O-methylwogonin 5-glucoside,  skullcapflavone I 2’-glucoside, neoandrographolide,  14-deoxy-11-hydroxyandro grapholide, 7-methoxy luteoline,  luteoline,

Triterpnoids:
β-amyrin,  lupeol,  glutinol

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